Publications

WAZYNSKA, M., R. BUTERA, M. REQUESENS, A. PLAT, T. ZARGANES-TZITZIKAS, C. NEOCHORITIS, J. PLEWKA, L. SKALNIAK, J. KOCIK-KROL, B. MUSIELAK, K. MAGIERA-MULARZ, I. RODRIGUEZ, S. BLOK, M. DE BRYUN, H. NIJMAN, P. ELSINGA, T. HOLAK, A. DÖMLING

Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors. Journal of Medicinal Chemistry. 2023, 66(14), 9577-9591, ISSN: 0022-2623, PMID: 37450644,

SHALDAM, M., D. HENDRYCHOVA, R. EL-HAGGAR, V. VOJÁČKOVÁ, T. MAJRASHI, E. ELKAEED, N. MASURIER, V. KRYŠTOF, H. TAWFIK, W. ELDEHNA

2,4-Diaryl-pyrimido[1,2-a]benzimidazole derivatives as novel anticancer agents endowed with potent anti-leukemia activity: Synthesis, biological evaluation and kinase profiling. European Journal of Medicinal Chemistry. 2023, 258, 115610, ISSN: 0223-5234, PMID: 37437350, PDF.

DVOŘÁKOVÁ BENDOVÁ, K., V. RACLAVSKÝ, R. NOVOTNY, D. LUPTAKOVA, M. POPPER, Z. NOVÝ, M. HAJDÚCH, M. PETŘÍK

[68Ga]Ga-Ornibactin for Burkholderia cepacia complex Infection Imaging Using Positron Emission Tomography. Journal of Medicinal Chemistry. 2023, ISSN: 0022-2623, PMID: 37252893,

DAS, V., M. HAJDÚCH

Randomizing for Alzheimer's disease drug trials should consider the cancer history of participants. Brain. 2023, ISSN: 0006-8950, PMID: 37243427, PDF.

KANELLIS, D., A. ZISI, Z. ŠKROTT, B. LEMMENS, J. ESPINOZA, M. KOSAR, A. BJÖRKMAN, X. LI, S. ARAMPATZIS, J. BARTKOVA, M. ANDUJAR-SANCHEZ, O. FERNANDEZ-CAPETILLO, M. MISTRÍK, M. LINDSTROM, J. BÁRTEK

Actionable cancer vulnerability due to translational arrest, p53 aggregation and ribosome biogenesis stress evoked by the disulfiram metabolite CuET. Cell Death and Differentiation. 2023, ISSN: 1350-9047, PMID: 37142656,

BUCHTOVÁ, T., L. BÉRESOVÁ, K. CHROMÁ, T. PLUHACEK, T. BERES, D. KACZOROVA, P. TARKOWSKI, J. BÁRTEK, M. MISTRÍK

Cannabis-derived products antagonize platinum drugs by altered cellular transport. Biomedicine & Pharmacotherapy. 2023, 163, 114801, ISSN: 0753-3322, PMID: 37137184, PDF.

IVASECHKO, I., A. LOZYNSKYI, J. SENKIV, P. ROSZCZENKO, Y. KOZAK, N. FINIUK, O. KLYUCHIVSKA, N. KASHCHAK, N. MANKO, Z. MASLYAK, D. LESYK, A. KARKHUT, S. POLOKVOVYCH, R. CZARNOMYSY, O. SZEWCZYK, A. KOZYTSKIY, O. KARPENKO, D. KHYLUK, A. GZELLA, K. BIELAWSKI, A. BIELAWSKA, P. DŽUBÁK, S. GURSKÁ, M. HAJDÚCH, R. STOIKA, R. LESYK

Molecular design, synthesis and anticancer activity of new thiopyrano[2,3-d]thiazoles based on 5-hydroxy-1,4-naphthoquinone (juglone). European Journal of Medicinal Chemistry. 2023, 252, 115304, ISSN: 0223-5234, PMID: 37001390, PDF.

KOVALOVA, M., J. BARAKA, V. MIK, R. JORDA, M. LUO, H. SHAO, V. KRYŠTOF

A patent review of cyclin-dependent kinase 7 (CDK7) inhibitors (2018-2022). Expert Opinion on Therapeutic Patents. 2023, 33(2), 67-87, ISSN: 1354-3776, PMID: 36975020, PDF.

NOVÁKOVÁ (ČARNÁ), M., I. ONYANGO, S. KATINA, D. HOLUB, J. NOVOTNÝ, M. NEZVEDOVA, D. JHA, Z. NEDELSKA, V. LACOVICH, T. VYVERE, R. HOUBRECHTS, K. GARCIA-MANSFIELD, R. SHARMA, V. DAVID-DIRGO, M. VYHNALEK, K. TEXLOVA, H. CHAVES, N. BAKKAR, L. PERTIERRA, M. VINKLER, H. MARKOVA, J. LACZO, K. SHEARDOVA, M. HORTOVA-KOHOUTKOVA, J. FRIC, G. FORTE, P. KANOVSKY, S. BELASKOVA, J. DAMBORSKY, J. HORT, N. SEYFRIED, R. BOWSER, G. SEVLEVER, R. RISSMAN, R. SMITH, M. HAJDÚCH, P. PIRROTTE, Z. SPACIL, E. DAMMER, C. LIMBACK-STOKIN, G. STOKIN

Pathogenesis of Alzheimer's disease: Involvement of the choroid plexus. Alzheimer's & Dementia : the Journal of the Alzheimer's Association. 2023, ISSN: 1552-5260, PMID: 36825691, PDF.

PERINA, M., M. KISS, G. MOTYAN, E. SZCZYRBOVA, M. ELIÁŠ, V. STUDENT, D. KURFÜRSTOVÁ, M. KOVALOVA, L. MADA, J. BOUCHAL, E. FRANK, R. JORDA

A-ring-fused pyrazoles of dihydrotestosterone targeting prostate cancer cells via the downregulation of the androgen receptor. European Journal of Medicinal Chemistry. 2023, 249, 115086, ISSN: 0223-5234, PMID: 36682291, PDF.

Publications

Published in Top 10% journals in the field